SCHEMBL290463

SCHEMBL290463

COCCCn1c(=O)oc2ccc(-c3ccc(C(C#N)CNC(=O)C4(NC(=O)O)CCOCC4)cc3)cc21

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSC P53634 14/20 0.49
KCNH2 Q12809 1/20 0.37
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
ASAH1 Q13510 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290107 0.96 CTSC (0.49) CTSCKCNH2SMN1; SMN2
SCHEMBL290320 0.87 CTSC (0.45) CTSCKCNH2
SCHEMBL2885392 0.86 CTSC (0.62) CTSCKCNH2
SCHEMBL290293 0.82 CTSC (0.50) CTSCKCNH2
SCHEMBL2890775 0.82 CTSC (0.62) CTSCKCNH2
SCHEMBL290462 0.80 CTSC (0.46) CTSCKCNH2MEN1NPC1TSHR
SCHEMBL299037 0.80 CTSC (0.49) CTSCKCNH2MEN1NPC1TSHR
SCHEMBL7871687 0.78 CTSC (0.59) CTSCKCNH2
SCHEMBL16478129 0.78 CTSC (0.52) CTSCKCNH2ASAH1MAPT
SCHEMBL16478115 0.78 CTSC (0.49) CTSCKCNH2ASAH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed