SCHEMBL2904958

SCHEMBL2904958

COC(=O)[C@@H]1[C@@H](O)CCN1CCN1CCN(C(=O)/C=C/c2ccc(Cl)c(Cl)c2)CCC1=O

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 8/20 0.45
GPR183 P32249 5/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
TDP1 Q9NUW8 1/20 0.43
SLC2A1 P11166 1/20 0.42
ALDH1A1 P00352 1/20 0.39
ITGB2 P05107 1/20 0.39
ICAM1 P05362 1/20 0.39
ITGAL P20701 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904960 1.00 CCR2 (0.45) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2897297 0.86 GPR183 (0.48) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2897296 0.86 GPR183 (0.48) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2899751 0.81 GPR183 (0.48) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2897826 0.81 NPC1 (0.51) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2903750 0.79 GPR183 (0.44) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2903753 0.79 GPR183 (0.44) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL1556326 0.79 NPC1 (0.53) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL1556324 0.79 NPC1 (0.53) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2903128 0.78 CCR2 (0.51) CCR2GPR183NPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed