SCHEMBL29055014

SCHEMBL29055014

COc1cc2c(N3CCCN(C(=O)O)CC3)ncnc2cc1O

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.64
BACE1 P56817 2/20 0.64
ENPP1 P22413 4/20 0.61
AURKA O14965 1/20 0.59
PDGFRB P09619 13/20 0.58
PDGFRA P16234 4/20 0.58
KIT P10721 1/20 0.53
FLT3 P36888 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23726540 0.87 TLR9 (0.65) ACHEBACE1ENPP1AURKAPDGFRB
SCHEMBL30080209 0.87 TLR9 (0.65) ACHEBACE1ENPP1AURKAPDGFRB
Hydrochloric Acid SCHEMBL2915718 0.86 ACHE (0.80) ACHEBACE1ENPP1AURKAPDGFRB
SCHEMBL4726710 0.84 ENPP1 (0.65) ACHEBACE1ENPP1AURKAPDGFRB
SCHEMBL22631414 0.83 ACHE (0.67) ACHEBACE1ENPP1AURKAPDGFRB
SCHEMBL29055085 0.83 PDGFRB (0.69) ACHEBACE1ENPP1AURKAPDGFRB
SCHEMBL25656495 0.83 ENPP1 (0.59) ACHEBACE1ENPP1AURKAPDGFRB
SCHEMBL23762347 0.83 ENPP1 (0.85) ACHEBACE1ENPP1AURKA
Hydrochloric Acid SCHEMBL23726065 0.82 ENPP1 (0.84) ACHEBACE1ENPP1AURKA
Hydrochloric Acid SCHEMBL30079993 0.82 ENPP1 (0.84) ACHEBACE1ENPP1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115362145-A Ecto-nucleotide pyrophosphatase/phosphodiesterase 1 (ENPP 1) inhibitors and methods of use thereof 斯汀格瑞治疗股份有限公司 2022-11-18 CN disclosed