SCHEMBL29055293

SCHEMBL29055293

COc1ccccc1C1=CCC(C(=O)Nc2cc(OCCN(C)C)c(C#N)cn2)(c2noc(C)n2)C=C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 14/20 0.42
HTR1D P28221 4/20 0.38
HTR1B P28222 4/20 0.38
HTR2A P28223 4/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTR7 P34969 2/20 0.37
CHRM2 P08172 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29055282 0.92 FGFR4 (0.42) FGFR4HTR1DHTR1BHTR2AKDM4E
SCHEMBL29055283 0.90 FGFR4 (0.41) FGFR4HTR1DHTR1BHTR2AKDM4E
SCHEMBL29055273 0.90 HTR1D (0.39) FGFR4HTR1DHTR1BHTR2AKDM4E
SCHEMBL29055285 0.88 FGFR4 (0.39) FGFR4HTR1DHTR1BHTR2AKDM4E
SCHEMBL29055280 0.81 HTR1D (0.35) FGFR4HTR1DHTR1BHTR2AKDM4E
SCHEMBL29055281 0.81 HTR1D (0.35) FGFR4HTR1DHTR1BHTR2AKDM4E
SCHEMBL29055294 0.80 RORC (0.33) FGFR4HTR1DHTR1BHTR2AKDM4E
SCHEMBL29055279 0.80 HTR1D (0.34) FGFR4HTR1DHTR1BHTR2AKDM4E
SCHEMBL29055287 0.80 RORC (0.33) FGFR4KDM4EALDH1A1HPGDHSD17B10
SCHEMBL29055292 0.79 CNR2 (0.34) S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116635390-A Potent and selective compounds as serotonin 1B receptor modulators 莱科斯生物技术公司 2023-08-22 CN claimed
CN-116635390-A Potent and selective compounds as serotonin 1B receptor modulators 莱科斯生物技术公司 2023-08-22 CN disclosed