SCHEMBL29058902

SCHEMBL29058902

CC(C)(C)OC(=O)c1ccc(N2CC(CN3CCN(C(=O)OCc4ccccc4)CC3)C2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 6/20 0.45
SIGMAR1 Q99720 6/20 0.45
PARP1 P09874 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
PDK1 Q15118 1/20 0.43
PDK2 Q15119 1/20 0.43
PDK3 Q15120 1/20 0.43
PDK4 Q16654 1/20 0.43
CYP2C19 P33261 1/20 0.42
CHRM4 P08173 2/20 0.42
CNR1 P21554 1/20 0.42
ESRRB O95718 1/20 0.41
ESR1 P03372 1/20 0.41
ESRRA P11474 1/20 0.41
ESRRG P62508 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28528615 0.92 GPR119 (0.47) TMEM97SIGMAR1MEN1KMT2ANPSR1
SCHEMBL29058862 0.88 TMEM97 (0.44) TMEM97SIGMAR1PARP1MEN1KMT2A
SCHEMBL25338897 0.84 SMN1; SMN2 (0.50) PARP1MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL20046470 0.84 SMN1; SMN2 (0.50) PARP1MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL31291575 0.82 KMT2A (0.52) SIGMAR1PARP1MEN1KMT2ANPSR1
SCHEMBL30179036 0.81 SMN1; SMN2 (0.53) PARP1SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL30602886 0.81 SMN1; SMN2 (0.53) PARP1SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL26705305 0.81 SMN1; SMN2 (0.53) PARP1SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL29132380 0.81 SMN1; SMN2 (0.54) PARP1MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL29579133 0.81 SMN1; SMN2 (0.49) PARP1MEN1KMT2ANPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010858-B BTK inhibitor, preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2023-07-18 CN disclosed
CN-112010858-A BTK inhibitor, preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-12-01 CN disclosed