SCHEMBL2907254

SCHEMBL2907254

O=C(O)c1cc(NCc2ccccn2)nc(-c2ccccc2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.56
ABCG2 Q9UNQ0 1/20 0.56
PTGS2 P35354 1/20 0.53
PDE5A O76074 2/20 0.52
RAB9A P51151 3/20 0.49
KDM4E B2RXH2 3/20 0.49
NPC1 O15118 2/20 0.49
LMNA P02545 2/20 0.49
POLB P06746 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 1/20 0.47
NAMPT P43490 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2909195 0.83 ABCB1 (0.52) ABCB1ABCG2PTGS2PDE5AKDM4E
SCHEMBL13309934 0.83 ABCB1 (0.62) ABCB1ABCG2PTGS2PDE5ARAB9A
SCHEMBL16392006 0.80 ABCG2 (0.79) ABCB1ABCG2PTGS2PDE5ARAB9A
SCHEMBL2907007 0.78 ABCB1 (0.58) ABCB1ABCG2PDE5ARAB9AKDM4E
SCHEMBL2905528 0.76 ABCG2 (0.44) ABCB1ABCG2NPC1KMT2AADORA2A
SCHEMBL12923510 0.76 MAPT (0.47) ABCB1ABCG2PDE5AKDM4ELMNA
SCHEMBL2903558 0.73 ADORA2A (0.54) KDM4ELMNAMAPK1KMT2AADORA2A
SCHEMBL27827798 0.73 ABCG2 (0.60) ABCB1ABCG2RAB9ANPC1KMT2A
SCHEMBL2905601 0.72 ADORA1 (0.45) PTGS2KMT2AADORA2AADORA1ALDH1A1
SCHEMBL27846476 0.71 SCN9A (0.55) KMT2AADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217606-A1 SOLUBILIZED THIAZOLOPYRIDINES Sirtris Pharmaceuticals, Inc. (US) 2010-08-18 EP disclosed
WO-2009061453-A1 SOLUBILIZED THIAZOLOPYRIDINES SIRTRIS PHARMACEUTICALS, INC. (US) 2009-05-14 WO disclosed