SCHEMBL2907007

SCHEMBL2907007

O=C(O)c1cc(NCc2cccnc2)nc(-c2ccccc2)n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.58
ABCC1 P33527 1/20 0.58
ABCG2 Q9UNQ0 1/20 0.58
CYP1A2 P05177 10/20 0.54
CYP3A4 P08684 10/20 0.54
CYP2D6 P10635 8/20 0.54
CYP2C19 P33261 7/20 0.54
CLK4 Q9HAZ1 6/20 0.54
ALOX15 P16050 2/20 0.54
ALDH1A1 P00352 7/20 0.54
PDE5A O76074 2/20 0.54
CYP2C9 P11712 2/20 0.54
POLB P06746 1/20 0.54
USP2 O75604 1/20 0.53
HPGD P15428 2/20 0.52
HSD17B10 Q99714 5/20 0.50
TSHR P16473 3/20 0.50
MAPK1 P28482 2/20 0.50
VNN1 O95497 1/20 0.50
KMT2A Q03164 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2909195 0.89 ABCB1 (0.52) ABCB1ABCG2CYP1A2CYP3A4CYP2D6
SCHEMBL2907254 0.78 ABCB1 (0.56) ABCB1ABCG2CLK4ALDH1A1PDE5A
SCHEMBL12923327 0.76 HPGD (0.52) ABCB1ABCC1ABCG2CYP1A2CYP3A4
SCHEMBL13188295 0.76 ABCB1 (0.48) ABCB1ABCC1ABCG2CYP1A2CYP3A4
SCHEMBL12923516 0.76 HPGD (0.47) ABCB1ABCC1ABCG2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL984560 0.76 HPGD (0.51) ABCB1ABCC1ABCG2CYP1A2CYP3A4
SCHEMBL3721157 0.76 ABCB1 (0.48) ABCB1ABCC1ABCG2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL985536 0.75 HPGD (0.47) ABCB1ABCC1ABCG2CYP1A2CYP3A4
SCHEMBL2905528 0.75 ABCG2 (0.44) ABCB1ABCC1ABCG2ALDH1A1KMT2A
SCHEMBL13309776 0.74 CYP3A4 (0.67) CYP1A2CYP3A4CYP2D6CYP2C19CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217606-A1 SOLUBILIZED THIAZOLOPYRIDINES Sirtris Pharmaceuticals, Inc. (US) 2010-08-18 EP disclosed
WO-2009061453-A1 SOLUBILIZED THIAZOLOPYRIDINES SIRTRIS PHARMACEUTICALS, INC. (US) 2009-05-14 WO disclosed