SCHEMBL29072952

SCHEMBL29072952

CC(C)COc1ccc(CNC(=O)N(Cc2ccc(F)cc2)C[C@H]2CCNC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 20/20 0.69
HTR2C P28335 4/20 0.58
ABCB11 O95342 1/20 0.58
CYP1A2 P05177 1/20 0.58
ADRB2 P07550 1/20 0.58
CHRM2 P08172 1/20 0.58
CHRM1 P11229 1/20 0.58
DRD1 P21728 1/20 0.58
TBXA2R P21731 1/20 0.58
SLC6A2 P23975 1/20 0.58
GPR183 P32249 1/20 0.58
CYP2C19 P33261 1/20 0.58
ADRA1A P35348 1/20 0.58
OPRM1 P35372 1/20 0.58
APLNR P35414 1/20 0.58
DRD3 P35462 1/20 0.58
CX3CR1 P49238 1/20 0.58
SLC6A3 Q01959 1/20 0.58
KCNH2 Q12809 1/20 0.58
GPR65 Q8IYL9 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29072954 1.00 HTR2A (0.69) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL28271149 0.92 HTR2A (0.57) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL28271150 0.92 HTR2A (0.57) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL29073202 0.85 HTR2A (0.59) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL23686881 0.85 HTR2A (0.74) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL23686824 0.84 HTR2A (0.48) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL23686868 0.84 HTR2A (0.66) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20765948 0.84 HTR2A (0.64) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20766182 0.84 HTR2A (0.64) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL23686966 0.84 HTR2A (0.70) HTR2AHTR2CABCB11CYP1A2ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109111385-B 5-HT 2A Receptor inhibitor and preparation method and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed