SCHEMBL2907585

SCHEMBL2907585

CCOC(=O)c1cnc2cc(OCC)c(Br)cc2c1Nc1cc(F)cc(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.54
CA2 P00918 1/20 0.51
TP53 P04637 2/20 0.50
GAA P10253 3/20 0.49
THRB P10828 1/20 0.49
CSF1R P07333 2/20 0.48
SMN1; SMN2 Q16637 4/20 0.47
LMNA P02545 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
AURKB Q96GD4 3/20 0.47
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.46
AURKA O14965 2/20 0.45
PAX8 Q06710 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912397 0.86 CA2 (0.61) MAPTCA2TP53GAATHRB
SCHEMBL2913228 0.86 MAPT (0.61) MAPTCA2TP53CSF1RSMN1; SMN2
SCHEMBL2908274 0.85 CA2 (0.61) MAPTCA2TP53GAATHRB
SCHEMBL2908202 0.85 CA2 (0.61) MAPTCA2TP53GAATHRB
SCHEMBL2907504 0.84 MAPT (0.56) MAPTCA2TP53GAATHRB
SCHEMBL2904906 0.83 MAPT (0.58) MAPTCA2TP53GAATHRB
SCHEMBL2911948 0.83 CSF1R (0.59) MAPTGAACSF1RSMN1; SMN2LMNA
SCHEMBL2913852 0.83 CSF1R (0.59) MAPTCA2TP53GAATHRB
SCHEMBL2910243 0.83 CSF1R (0.59) MAPTCA2TP53GAATHRB
SCHEMBL2912285 0.83 CSF1R (0.58) MAPTCA2TP53GAATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed