SCHEMBL2907603

SCHEMBL2907603

CCc1ccc(-c2cn(CCCNc3ccc([N+](=O)[O-])c(N)n3)cc2NC(=O)C(CCCNC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.35
CA1 P00915 3/20 0.35
BRD4 O60885 1/20 0.33
BCL2 P10415 1/20 0.33
IDO1 P14902 2/20 0.32
HDAC4 P56524 3/20 0.32
HDAC1 Q13547 3/20 0.32
HDAC3 O15379 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912738 0.92 BCL2 (0.32) BCL2HDAC4HDAC1
SCHEMBL2909660 0.91 BCL2 (0.33) BCL2IDO1
SCHEMBL2907410 0.88 GSK3B (0.34)
SCHEMBL2910107 0.86 GSK3B (0.42) CA2CA1BRD4BCL2IDO1
SCHEMBL2904688 0.82 GSK3B (0.34)
SCHEMBL2905411 0.81 GSK3B (0.35)
SCHEMBL2912527 0.81 GSK3B (0.36)
SCHEMBL2910071 0.80 GSK3A (0.32)
SCHEMBL2912926 0.80 BDKRB1 (0.34)
SCHEMBL2908407 0.79 GSK3B (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed