SCHEMBL29092174

SCHEMBL29092174

C[S+]([O-])c1nc(Nc2ccc(N3CCOCC3)cc2)cc(N2CCN(C=O)CC2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 2/20 0.46
AURKA O14965 3/20 0.45
MAPT P10636 4/20 0.42
MAPK1 P28482 2/20 0.42
TP53 P04637 1/20 0.42
PLK4 O00444 1/20 0.41
GALR2 O43603 1/20 0.41
GALR1 P47211 1/20 0.41
ZAP70 P43403 1/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
PTK2B Q14289 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM1A O60341 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPK10 P53779 1/20 0.38
JAK2 O60674 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29091968 0.82 MAPT (0.49) IGF1RAURKAMAPTMAPK1TP53
SCHEMBL25386738 0.76 MAPK10 (0.41) AURKAMAPTTP53GALR2GALR1
SCHEMBL25386961 0.69 RAF1 (0.47) IGF1RMAPTMAPK1PLK4LMNA
SCHEMBL1124059 0.68 HTT (0.52) MAPTMAPK1LMNAALDH1A1GAA
SCHEMBL25387217 0.67 FYN (0.45) MAPTMAPK1TP53LMNAALDH1A1
SCHEMBL25388213 0.67 MAPT (0.44) MAPTGAAMEN1KMT2A
SCHEMBL5380919 0.66 KMT2A (0.50) IGF1RAURKAMAPTMAPK1TP53
SCHEMBL27875709 0.65 AURKA (0.66) AURKAMAPTMAPK1LMNAALDH1A1
SCHEMBL5402668 0.65 AURKA (0.48) IGF1RAURKAMAPTMAPK1TP53
SCHEMBL12562997 0.65 PIK3CB (0.46) MAPTMAPK1ALDH1A1GAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116507611-A Novel capsid assembly inhibitor 佩勒梅德有限公司 2023-07-28 CN claimed
CN-116507611-A Novel capsid assembly inhibitor 佩勒梅德有限公司 2023-07-28 CN disclosed