SCHEMBL2909714

SCHEMBL2909714

Nc1nc(NCCCn2cc(C(=O)O)c(-c3ccc(Br)cc3)c2)ccc1[N+](=O)[O-]

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.36
GSK3A P49840 3/20 0.36
EIF4E P06730 1/20 0.35
LMNA P02545 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
CDK1 P06493 2/20 0.34
FOLH1 Q04609 1/20 0.33
CCNB2 O95067 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
SIRT5 Q9NXA8 2/20 0.33
DHFR P00374 1/20 0.32
CDK2 P24941 1/20 0.31
MEN1 O00255 2/20 0.31
MAPT P10636 2/20 0.31
HTT P42858 2/20 0.31
KMT2A Q03164 2/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2911792 0.91 GSK3B (0.36) GSK3BGSK3AEIF4ELMNACDK1
SCHEMBL2907084 0.91 GSK3B (0.37) GSK3BGSK3AEIF4ELMNACDK1
SCHEMBL2904891 0.91 GSK3B (0.42) GSK3BGSK3AEIF4ELMNACDK1
SCHEMBL2904612 0.90 GSK3B (0.36) GSK3BGSK3ACDK1FOLH1CCNB2
SCHEMBL2911406 0.89 EIF4E (0.37) GSK3BGSK3AEIF4ELMNACDK1
SCHEMBL2912610 0.89 MAPT (0.38) GSK3BGSK3AEIF4ELMNAMAPT
SCHEMBL2905948 0.89 EIF4E (0.37) GSK3BGSK3AEIF4ECDK1FOLH1
SCHEMBL2908029 0.87 GSK3B (0.37) GSK3BGSK3AEIF4ELMNACYP1A2
SCHEMBL2911906 0.87 CYP1A2 (0.34) GSK3BGSK3ALMNACYP1A2CYP2C19
SCHEMBL2904664 0.87 CYP1A2 (0.34) GSK3BGSK3ALMNACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed