SCHEMBL2909822

SCHEMBL2909822

Cc1onc(-c2ccccc2)c1CNC(=O)c1cn(CCCNc2ccc([N+](=O)[O-])c(N)n2)cc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.43
GSK3A P49840 3/20 0.43
CDK1 P06493 2/20 0.40
CCNB2 O95067 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
ALDH1A1 P00352 4/20 0.39
MAPT P10636 3/20 0.39
PLA2G1B P04054 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
GABRA5 P31644 4/20 0.36
ENPP2 Q13822 1/20 0.36
KDM4E B2RXH2 1/20 0.35
AKR1C3 P42330 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
PKM P14618 1/20 0.34
HTT P42858 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2909753 0.86 HPGD (0.47) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2910286 0.83 GSK3B (0.43) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2904121 0.82 GSK3B (0.44) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2904086 0.82 HPGD (0.45) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2909523 0.82 GSK3B (0.48) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2911606 0.82 GSK3B (0.48) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2904255 0.82 GSK3B (0.47) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2912130 0.81 GSK3B (0.48) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2910338 0.81 GSK3B (0.45) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2911627 0.81 GSK3B (0.46) GSK3BGSK3ACDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed