SCHEMBL2911041

SCHEMBL2911041

CCOc1cc2ncc(C(N)=O)c(Nc3ccc(F)c(Cl)c3)c2cc1N1CCN(C2CC2)CC1

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 15/20 0.61
KCNH2 Q12809 5/20 0.60
SCN5A Q14524 3/20 0.60
EGFR P00533 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913453 0.91 CSF1R (0.73) CSF1RKCNH2SCN5A
SCHEMBL2904777 0.90 CSF1R (0.64) CSF1RKCNH2SCN5AEGFR
SCHEMBL2910817 0.89 CSF1R (0.63) CSF1RKCNH2SCN5AEGFR
SCHEMBL2904770 0.89 CSF1R (0.65) CSF1RKCNH2SCN5AEGFR
SCHEMBL2910284 0.89 CSF1R (0.62) CSF1RKCNH2SCN5AEGFR
SCHEMBL2910987 0.88 KCNH2 (0.74) CSF1RKCNH2SCN5A
SCHEMBL2909948 0.88 CSF1R (0.73) CSF1RKCNH2SCN5A
SCHEMBL2913641 0.87 CSF1R (0.65) CSF1RKCNH2SCN5AEGFR
SCHEMBL2907894 0.87 KCNH2 (0.71) CSF1RKCNH2SCN5A
SCHEMBL28780792 0.86 CSF1R (0.60) CSF1RKCNH2SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed
CN-101466682-A 4-anilinoquinolina-3-carboxamidas como inhibidores de la quinasa CSF-1R ASTRAZENECA AB (SE) 2009-06-24 CN disclosed