SCHEMBL29119613

SCHEMBL29119613

CC(C)(C)OC(=O)n1cc(Br)c(B(O)O)n1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.33
BCHE P06276 1/20 0.32
HTT P42858 1/20 0.32
ATM Q13315 1/20 0.32
KDM1A O60341 1/20 0.31
FAAH O00519 1/20 0.31
ELANE P08246 1/20 0.31
SCD O00767 1/20 0.31
LMNA P02545 1/20 0.30
GPR119 Q8TDV5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL481939 0.81 ROCK2 (0.34) ROCK2BCHEHTTATMFAAH
SCHEMBL18603273 0.79 KCNH2 (0.34) ROCK2BCHEHTTATMFAAH
SCHEMBL4699798 0.79 ROCK2 (0.36) ROCK2BCHEHTTATMFAAH
SCHEMBL30771246 0.79 AR (0.34) ROCK2BCHEHTTATMFAAH
SCHEMBL23751758 0.76 HTT (0.37) ROCK2HTTATMGPR119
SCHEMBL581742 0.76 KCNH2 (0.35) ROCK2HTTATMGPR119
SCHEMBL18387648 0.75 EPHX2 (0.47) ROCK2HTTELANEGPR119
SCHEMBL28574885 0.75 ROCK2 (0.34) ROCK2BCHE
Boric Acid SCHEMBL29391967 0.72 ELANE (0.44) ROCK2BCHEHTTATMELANE
SCHEMBL17631624 0.71 HDAC8 (0.39) ROCK2BCHEHTTKDM1ASCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112930348-B Improved process for the manufacture of 3- [ (1S) -1-imidazo [1,2-a ] pyridin-6-ylethyl ] -5- (1-methylpyrazol-4-yl) triazolo [4,5-b ] pyrazines and polymorphic forms thereof 阿斯利康(瑞典)有限公司 2023-12-05 CN disclosed