SCHEMBL2912205

SCHEMBL2912205

Nc1nc(NCCCn2cc(-c3ccc(Cl)cc3Cl)cc2C(=O)NCCCN2CCCC2)ccc1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.49
GSK3A P49840 3/20 0.49
CDK1 P06493 2/20 0.43
LMNA P02545 2/20 0.43
CCNB2 O95067 1/20 0.43
CCNB1 P14635 1/20 0.43
CCNB3 Q8WWL7 1/20 0.43
CACNA1G O43497 2/20 0.39
MAPT P10636 2/20 0.39
KLK7 P49862 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
MCHR1 Q99705 1/20 0.38
CYP2C19 P33261 1/20 0.37
F10 P00742 1/20 0.37
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2907104 0.97 GSK3B (0.49) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL2911669 0.94 LMNA (0.53) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL2911942 0.91 CYP2C19 (0.50) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL2913436 0.90 GSK3B (0.48) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL13211506 0.90 GSK3B (0.43) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL2911878 0.88 GSK3B (0.48) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL2914191 0.88 GSK3B (0.47) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL2904013 0.87 GSK3B (0.52) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL2903944 0.87 GSK3B (0.51) GSK3BGSK3ACDK1LMNACCNB2
SCHEMBL2907721 0.87 GSK3B (0.49) GSK3BGSK3ACDK1LMNACCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed