SCHEMBL2912246

SCHEMBL2912246

CCOC(=O)c1cnc2cc(OCC)c(N3CCCN(C)CC3)cc2c1Nc1ccc(F)c(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.62
SCN5A Q14524 3/20 0.58
CSF1R P07333 10/20 0.57
GAA P10253 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
SLC2A1 P11166 1/20 0.52
MAPT P10636 2/20 0.51
EGFR P00533 2/20 0.51
CA2 P00918 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2905235 0.97 KCNH2 (0.61) KCNH2SCN5ACSF1RGAAMEN1
SCHEMBL2907516 0.94 CSF1R (0.60) KCNH2SCN5ACSF1RGAAMEN1
SCHEMBL2911379 0.93 CSF1R (0.66) KCNH2SCN5ACSF1RGAAMEN1
SCHEMBL2910987 0.92 KCNH2 (0.74) KCNH2SCN5ACSF1R
SCHEMBL2909956 0.91 KCNH2 (0.61) KCNH2SCN5ACSF1RGAAMEN1
SCHEMBL2911915 0.90 GAA (0.53) KCNH2SCN5ACSF1RGAAMAPT
SCHEMBL2911202 0.90 CSF1R (0.70) KCNH2SCN5ACSF1RGAAMEN1
SCHEMBL2913652 0.90 CSF1R (0.57) KCNH2SCN5ACSF1RGAAMEN1
SCHEMBL2910871 0.89 MAPT (0.64) KCNH2SCN5ACSF1RGAAMEN1
SCHEMBL2911172 0.89 MAPT (0.52) KCNH2SCN5ACSF1RGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed