SCHEMBL2910871

SCHEMBL2910871

CCOC(=O)c1cnc2cc(OCC)c(N3CCOCC3)cc2c1Nc1ccc(F)c(Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.64
GAA P10253 8/20 0.64
SMN1; SMN2 Q16637 3/20 0.59
TDP1 Q9NUW8 3/20 0.59
L3MBTL1 Q9Y468 3/20 0.59
LMNA P02545 2/20 0.59
MC4R P32245 2/20 0.59
HTT P42858 2/20 0.59
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
PTK2B Q14289 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
MAPK1 P28482 2/20 0.59
CLK1 P49759 1/20 0.59
GSK3A P49840 1/20 0.59
GSK3B P49841 1/20 0.59
TP53 P04637 1/20 0.57
EGFR P00533 4/20 0.56
CSF1R P07333 1/20 0.53
CA2 P00918 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912890 0.93 MAPT (0.65) MAPTGAASMN1; SMN2TDP1L3MBTL1
SCHEMBL2905235 0.92 KCNH2 (0.61) MAPTGAAMEN1KMT2AEGFR
SCHEMBL2911915 0.92 GAA (0.53) MAPTGAAEGFRCSF1RCA2
SCHEMBL2904770 0.91 CSF1R (0.65) EGFRCSF1RKCNH2SCN5A
SCHEMBL2911172 0.90 MAPT (0.52) MAPTGAASMN1; SMN2TDP1L3MBTL1
SCHEMBL2912246 0.89 KCNH2 (0.62) MAPTGAAMEN1KMT2AEGFR
SCHEMBL2907516 0.89 CSF1R (0.60) MAPTGAAMEN1KMT2AEGFR
SCHEMBL2907899 0.88 CSF1R (0.55) MAPTGAAEGFRCSF1RCA2
SCHEMBL2911375 0.88 CSF1R (0.66) MAPTGAASMN1; SMN2TDP1L3MBTL1
SCHEMBL2912768 0.88 CA2 (0.51) MAPTGAASMN1; SMN2TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed