SCHEMBL2912637

SCHEMBL2912637

Nc1nc(NCCCn2cc(C(=O)NCCc3cccnc3)c(-c3ccc(Cl)cc3Cl)c2)ccc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
GSK3B P49841 5/20 0.46
GSK3A P49840 3/20 0.46
CDK1 P06493 2/20 0.46
HTT P42858 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
DPP4 P27487 1/20 0.44
DPP8 Q6V1X1 1/20 0.44
DPP9 Q86TI2 1/20 0.44
CCNB2 O95067 1/20 0.44
CCNB1 P14635 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CDK5 Q00535 1/20 0.40
CDK5R1 Q15078 1/20 0.40
MAPT P10636 2/20 0.39
HDAC8 Q9BY41 1/20 0.39
PTAFR P25105 2/20 0.38
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2903991 0.94 POLB (0.56) POLBGSK3BGSK3ACDK1HTT
SCHEMBL2907243 0.92 GSK3B (0.46) POLBGSK3BGSK3ACDK1SMN1; SMN2
SCHEMBL2909753 0.87 HPGD (0.47) POLBGSK3BGSK3ACDK1HTT
SCHEMBL2911606 0.87 GSK3B (0.48) POLBGSK3BGSK3ACDK1HTT
SCHEMBL2909523 0.87 GSK3B (0.48) POLBGSK3BGSK3ACDK1HTT
SCHEMBL2912731 0.87 GSK3B (0.45) POLBGSK3BGSK3ACDK1SMN1; SMN2
SCHEMBL2904255 0.87 GSK3B (0.47) POLBGSK3BGSK3ACDK1HTT
SCHEMBL2910223 0.86 GSK3B (0.48) POLBGSK3BGSK3ACDK1SMN1; SMN2
SCHEMBL2911549 0.86 GSK3B (0.47) POLBGSK3BGSK3ACDK1HTT
SCHEMBL2910340 0.86 GSK3B (0.53) GSK3BGSK3ACDK1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed