SCHEMBL29129286

SCHEMBL29129286

Nc1nccc2ccc(-c3ccncc3)cc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 3/20 0.58
JAK2 O60674 1/20 0.51
F12 P00748 2/20 0.48
PLAU P00749 2/20 0.48
NCF1 P14598 1/20 0.48
NOS3 P29474 1/20 0.48
NOS1 P29475 1/20 0.48
NOS2 P35228 1/20 0.48
BACE1 P56817 1/20 0.48
MAPK10 P53779 1/20 0.48
PDPK1 O15530 2/20 0.47
AAK1 Q2M2I8 1/20 0.47
PRKCZ Q05513 1/20 0.46
PLG P00747 2/20 0.44
F11 P03951 1/20 0.44
KLKB1 P03952 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
PRSS3 P35030 1/20 0.44
PIK3CA P42336 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29987075 0.83 MAP4K4 (0.63) MAP4K4F12PLAUNCF1NOS3
SCHEMBL27990709 0.77 MAP4K4 (0.60) MAP4K4F12PLAUNCF1NOS3
SCHEMBL29508479 0.75 F12 (0.57) MAP4K4F12PLAUNCF1NOS3
SCHEMBL5989271 0.75 F12 (0.57) MAP4K4F12PLAUNCF1NOS3
SCHEMBL15587570 0.74 MAP4K4 (1.00) MAP4K4
SCHEMBL30834093 0.73 KDM4E (0.40) MAP4K4JAK2F12PLAUNCF1
SCHEMBL27201388 0.73 KDM4E (0.40) MAP4K4JAK2F12PLAUNCF1
SCHEMBL30834158 0.73 MAP4K4 (0.41) MAP4K4JAK2F12PLAUNCF1
SCHEMBL27201289 0.73 MAP4K4 (0.41) MAP4K4JAK2F12PLAUNCF1
SCHEMBL27201611 0.73 CLK1 (0.55) MAP4K4JAK2PIK3CAMAPTDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117279896-A Amino substituted pyrido ring compounds, preparation method and application thereof 劲方医药科技(上海)有限公司 2023-12-22 CN disclosed
WO-2022214044-A1 AMINE-SUBSTITUTED PYRIDINE FUSED RING COMPOUNDS, PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2022-10-13 WO disclosed