Lidocaine

Lidocaine

SCHEMBL29130

CCN(CC)CC(=O)Nc1c(C)cccc1C.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9A

The experimentally established mechanism targets of Lidocaine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN3A known ✓ Q9NY46 3/20 0.97
SCN4A known ✓ P35499 1/20 0.97
SCN5A known ✓ Q14524 1/20 0.97
SCN9A known ✓ Q15858 1/20 0.97
SCN1A known ✓ P35498 2/20 0.55
SCN2A known ✓ Q99250 2/20 0.55
MAPT P10636 4/20 1.00
LMNA P02545 3/20 1.00
BLM P54132 2/20 1.00
GAA P10253 2/20 1.00
ALDH1A1 P00352 3/20 0.97
CYP3A4 P08684 1/20 0.97
MAPK1 P28482 1/20 0.97
MC4R P32245 1/20 0.97
MC3R P41968 1/20 0.97
HTR3A P46098 1/20 0.97
HPGD P15428 3/20 0.71
TSHR P16473 2/20 0.66
RAB9A P51151 1/20 0.66
MEN1 O00255 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lidocaine SCHEMBL5159066 1.00 MAPT (1.00) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL9113024 1.00 MAPT (1.00) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL29128 0.98 MAPT (0.97) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL20599347 0.98 MAPT (0.97) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL27387919 0.98 MAPT (0.97) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL5334354 0.98 MAPT (1.00) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL8183082 0.98 MAPT (1.00) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL15689 0.98 MAPT (1.00) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL28193323 0.97 MAPT (0.94) MAPTLMNABLMGAASCN3A
Lidocaine SCHEMBL28193322 0.97 MAPT (0.94) MAPTLMNABLMGAASCN3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 20061 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122075865-A Airway management apparatus with local anesthetic film and application thereof 2026-05-26 CN claimed
CN-122080445-A Sodium hyaluronate gel and preparation method thereof 2026-05-26 CN claimed
CN-122057064-A Multifunctional composite hemostatic powder capable of achieving wound in-situ self-gelation and preparation method thereof 杨鑫 2026-05-19 CN claimed
CN-122031677-A Leptin receptor agonist antibodies for the treatment of metabolic dysfunction or hypoleptinemia 瑞泽恩制药公司 2026-05-15 CN claimed
CN-122005915-A Antibiotic bioactive glass and preparation method thereof 山东秒亿通医学科技有限公司 2026-05-12 CN claimed
EP-4731182-A1 TOPICAL REGIMEN FOR TREATING COLD SORES Haleon UK IP Limited (GB) 2026-04-29 EP claimed
EP-4731181-A1 TOPICAL COMPOSITIONS FOR TREATING COLD SORES Haleon UK IP Limited (GB) 2026-04-29 EP claimed
EP-3723819-B1 WOUND DRESSING ANIMAL ETHICS PTY LTD (AU) 2026-04-22 EP claimed
US-20260097044-A1 ION PAIR LIQUID CRYSTAL FORMULATIONS FOR LONG-ACTING INJECTABLES OF POORLY SOLUBLE DRUGS FORDOZ PHARMA CORP. (US) 2026-04-09 US claimed
US-20260076872-A1 POLYMER VIALS WITH SUBSTANTIALLY FLAT BOTTOMS AND INJECTION STRETCH BLOW MOLDING METHODS FOR MAKING THE SAME SIO2 MEDICAL PRODUCTS LLC (US) 2026-03-19 US claimed
US-4439184-A Two-dose syringe CONCORD LABORATORIES, INC. (US) 1984-03-27 US claimed
US-4432758-A Urethral anesthetic devices FINEGOLD AARON N 1984-02-21 US claimed
US-4406883-A SHAPES MERRELL DOW PHARMACEUTICALS INC. (US) 1983-09-27 US claimed
EP-0060451-A1 Iontophoretic electrode MEDTRONIC, INC. (US) 1982-09-22 EP claimed
US-4339452-A ANTICOAGULANTS MEDICHEMIE AG (CH) 1982-07-13 US claimed
US-4312865-A Medication having penetration through cutaneous surfaces into articular and muscular areas SZUCS MURRILL M 1982-01-26 US claimed
US-4292300-A METHYL CELLULOSE, WATER, DRUG INVERESK RESEARCH INTERNATIONAL (GB) 1981-09-29 US claimed
US-4265875-A HYDROXYPROPYL METHYL CELLULOSE INVERESK RESEARCH INTERNATIONAL (GB) 1981-05-05 US claimed
US-4213876-A Multi-purpose blood diluent for use in electronic blood analysis instrumentation COULTER ELECTRONICS, INC. (US) 1980-07-22 US claimed
US-4091090-A PENETRANT ACCELERATOR COMPRISING CYCLOHEXYL-SUBSTITUTED ALKANOLS JOHNSON & JOHNSON (US) 1978-05-23 US claimed