SCHEMBL29131003

SCHEMBL29131003

Clc1ccc2c(n1)CCN(C1COC1)C2

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATR Q13535 10/20 0.39
HTR6 P50406 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
MAP4K1 Q92918 1/20 0.33
ABHD6 Q9BV23 1/20 0.33
GRM5 P41594 2/20 0.32
PDCD1LG2 Q9BQ51 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
PDE1B Q01064 1/20 0.31
KCNH2 Q12809 1/20 0.31
CYP3A4 P08684 1/20 0.31
MTOR P42345 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30602455 1.00 ATR (0.39) ATRHTR6HTR2AHTR2CHTR2B
SCHEMBL1507178 0.84 GRM5 (0.38) HTR2AHTR2CHTR2BCHRNB2CHRNA4
SCHEMBL15492555 0.82 PDE10A (0.41) ATRGRM5CD274CYP3A4MTOR
SCHEMBL28106897 0.80 KDR (0.42) HTR2AHTR2CHTR2BCHRNB2CHRNA4
SCHEMBL23554566 0.79 ATR (0.38) ATRHTR2AHTR2CHTR2BGRM5
SCHEMBL10255143 0.79 ATR (0.38) ATRGRM5CYP3A4MTOR
SCHEMBL23733445 0.79 ATR (0.38) ATRHTR6KCNH2CYP3A4MTOR
SCHEMBL31278237 0.77 ATR (0.37) ATRGRM5CYP3A4MTOR
SCHEMBL28835263 0.76 ABHD6 (0.39) ABHD6GRM5KCNH2
SCHEMBL31226154 0.75 PDE10A (0.39) ATRHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024245156-A1 HETEROCYCLIC COMPOUND ACTING AS α5-GABAA RECEPTOR REGULATOR 武汉人福创新药物研发中心有限公司 2024-12-05 WO disclosed
CN-119019425-A Alpha 5-GABAAHeterocyclic compounds as receptor modulators 武汉人福创新药物研发中心有限公司 2024-11-26 CN disclosed
CN-117069724-A Fused ring compounds, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-17 CN disclosed