SCHEMBL2913123

SCHEMBL2913123

CN1CCC[N]CC1CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
CHRNB2 P17787 1/20 0.33
CHRNA5 P30532 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
OPRD1 P41143 1/20 0.32
FFAR1 O14842 3/20 0.32
CHRM3 P20309 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2915892 0.89 TSHR (0.37) TSHROPRD1
SCHEMBL2912299 0.82 BRD4 (0.36) CHRNB2CHRNA5CHRNA7CHRNA4CHRM3
SCHEMBL2911063 0.82
SCHEMBL2919711 0.80 POLB (0.35) CHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL2918396 0.78 CYP1A2 (0.32)
SCHEMBL14077882 0.76 CHRNB2 (0.47) CHRNB2CHRNA5CHRNA7CHRNA4OPRD1
SCHEMBL13740779 0.76 CHRNB2 (0.47) CHRNB2CHRNA5CHRNA7CHRNA4OPRD1
SCHEMBL8198672 0.76 CHRNB2 (0.47) CHRNB2CHRNA5CHRNA7CHRNA4OPRD1
SCHEMBL2916570 0.75 CYP1A2 (0.34)
SCHEMBL2921981 0.74 CYP1A2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2734573-B1 BIODEGRADABLE, SEMI-CRYSTALLINE, PHASE SEPARATED, THERMOPLASTIC MULTI BLOCK COPOLYMERS FOR CONTROLLED RELEASE OF BIOLOGICALLY ACTIVE COMPOUNDS INNOCORE TECH HOLDING B V (NL) 2021-09-08 EP claimed
EP-2859887-B1 BIODEGRADABLE PHASE SEPARATED SEGMENTED MULTI BLOCK CO-POLYMERS AND RELEASE OF BIOLOGICALLY ACTIVE POLYPEPTIDES INNOCORE TECH B V (NL) 2017-03-22 EP claimed
EP-1709103-B1 BIODEGRADABLE MULTI-BLOCK CO-POLYMERS INNOCORE TECHNOLOGIES B V (NL) 2016-07-20 EP claimed
EP-1551899-B1 BIODEGRADABLE PHASE SEPARATED SEGMENTED MULTI BLOCK CO-POLYMERS INNOCORE TECHNOLOGIES B V (NL) 2008-05-07 EP claimed
EP-2225341-A1 METHOD FOR PRODUCING HYDROXY-FUNCTIONAL POLYMERS, THE ISOCYANATE-GROUP-TERMINATED POLYADDITION PRODUCTS WHICH CAN BE OBTAINED THEREFROM, AND THE USE THEREOF Sika Technology AG (CH) 2010-09-08 EP disclosed
EP-2143745-B1 Hybrid-functional polymers SIKA TECHNOLOGY AG (CH) 2010-04-21 EP disclosed
WO-2010003708-A1 HYBRID-FUNCTIONAL POLYMERS SIKA TECHNOLOGY AG (CH) 2010-01-14 WO disclosed
EP-2143745-A1 Hybrid-functional polymers Sika Technology AG (CH) 2010-01-13 EP disclosed
WO-2009077470-A1 METHOD FOR PRODUCING HYDROXY-FUNCTIONAL POLYMERS, THE ISOCYANATE-GROUP-TERMINATED POLYADDITION PRODUCTS WHICH CAN BE OBTAINED THEREFROM, AND THE USE THEREOF SIKA TECHNOLOGY AG (CH) 2009-06-25 WO disclosed
EP-2072556-A1 Method for creating hydroxyfunctional polymers, the isocyanate group terminal polyaddition products which can be gathered from them and their production Sika Technology AG (CH) 2009-06-24 EP disclosed