SCHEMBL29132897

SCHEMBL29132897

Cn1nccc1C1=C(N)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
COMT P21964 1/20 0.46
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
PI4KA P42356 1/20 0.41
PIK3CG P48736 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALOX5AP P20292 1/20 0.36
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
CDC42BPB Q9Y5S2 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15950989 0.77 COMT (0.60) COMTPIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL30060833 0.72 CYP1A2 (0.46) COMTPIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL16826278 0.71 CYP3A4 (0.53) COMTPIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL16877063 0.69 HSP90AA1 (0.46) COMTALDH1A1MAPTKDM4ENPC1
SCHEMBL31148179 0.68 COMT (0.43) COMTPIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL308138 0.67
SCHEMBL18985917 0.67 PIK3CD (0.55) COMTPIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL18518468 0.67 PIK3CD (0.48) COMTPIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL19462917 0.66 ALDH1A1 (0.41) COMTPIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL17796572 0.66 CYP1A2 (0.47) COMTPIK3CDPIK3CAPIK3CBPI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117304130-A MCL-1 inhibitors 吉利德科学公司 2023-12-29 CN disclosed
CN-112118845-B MCL-1 inhibitors 吉利德科学公司 2023-06-13 CN disclosed