SCHEMBL29132969

SCHEMBL29132969

COC1CN(C(=O)OC(C)(C)C)C1C

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
NR1H2 P55055 1/20 0.38
TSHR P16473 1/20 0.37
USP2 O75604 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.35
HPGD P15428 1/20 0.34
HSD11B1 P28845 1/20 0.34
CCR2 P41597 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29132972 1.00 CHRM2 (0.41) CHRM2CHRM1CHRM3NR1H2TSHR
SCHEMBL32664209 1.00 CHRM2 (0.41) CHRM2CHRM1CHRM3NR1H2TSHR
SCHEMBL21576380 1.00 CHRM2 (0.41) CHRM2CHRM1CHRM3NR1H2TSHR
SCHEMBL24070656 0.83 CHRM2 (0.42) CHRM2CHRM1CHRM3USP2SMN1; SMN2
SCHEMBL28923136 0.83 CHRM2 (0.42) CHRM2CHRM1CHRM3USP2SMN1; SMN2
SCHEMBL25698997 0.83 CHRM2 (0.42) CHRM2CHRM1CHRM3USP2SMN1; SMN2
SCHEMBL30867239 0.81 CHRM2 (0.38) CHRM2CHRM1CHRM3NR1H2USP2
SCHEMBL21227876 0.81 NR1H2 (0.42) CHRM2CHRM1CHRM3NR1H2TSHR
SCHEMBL27319966 0.81 NR1H2 (0.42) CHRM2CHRM1CHRM3NR1H2TSHR
SCHEMBL21227880 0.80 CHRM2 (0.37) CHRM2CHRM1CHRM3NR1H2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117304130-A MCL-1 inhibitors 吉利德科学公司 2023-12-29 CN disclosed
CN-112118845-B MCL-1 inhibitors 吉利德科学公司 2023-06-13 CN disclosed