SCHEMBL29132991

SCHEMBL29132991

COc1cc(-c2nnc(C)o2)c(F)cc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.47
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 4/20 0.38
HPGD P15428 4/20 0.38
HSD17B10 Q99714 3/20 0.38
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 2/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
BRD4 O60885 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
ACHE P22303 1/20 0.36
BACE1 P56817 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TSHR P16473 1/20 0.35
NOTUM Q6P988 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21958452 0.86 LRRK2 (0.48) LRRK2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL15651102 0.84 LRRK2 (0.47) LRRK2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL23997107 0.81 LRRK2 (0.45) LRRK2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL23997032 0.81 LRRK2 (0.48) LRRK2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL29133190 0.80 BRD4 (0.36) LRRK2BRD4CA12CA1CA2
SCHEMBL29133171 0.79 TP53 (0.42) LRRK2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL29132966 0.75 CA2 (0.36) LRRK2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL30622260 0.75 CA2 (0.36) LRRK2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL15272014 0.74 KDM4E (0.52) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL30622155 0.74 KDM4E (0.52) ALDH1A1KDM4EHPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed