SCHEMBL29133089

SCHEMBL29133089

COCc1cc(C(=O)NN)ccc1Br

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.53
CYP3A4 P08684 2/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
MAPT P10636 6/20 0.49
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
OGG1 O15527 1/20 0.47
MPO P05164 1/20 0.44
KDM5A P29375 1/20 0.44
BLM P54132 1/20 0.44
GFER P55789 1/20 0.44
PMP22 Q01453 1/20 0.44
HIF1A Q16665 1/20 0.44
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133080 0.85 TP53 (0.41) ALDH1A1CYP3A4MEN1KMT2ACYP1A2
SCHEMBL30622268 0.84 NOTUM (0.50) ALDH1A1CYP3A4MEN1KMT2ACYP1A2
SCHEMBL256771 0.84 NOTUM (0.50) ALDH1A1CYP3A4MEN1KMT2ACYP1A2
SCHEMBL24595665 0.82 ALDH1A1 (0.48) ALDH1A1MEN1KMT2AMAPTGAA
SCHEMBL30622253 0.82 ALDH1A1 (0.48) ALDH1A1MEN1KMT2AMAPTGAA
SCHEMBL408849 0.82 CA1 (0.44) ALDH1A1CA1CA2KDM5ARAB9A
SCHEMBL29133180 0.79 GSK3B (0.49) ALDH1A1MEN1KMT2AMAPTGAA
SCHEMBL30602390 0.78 ALDH1A1 (0.42) ALDH1A1MEN1KMT2ASMN1; SMN2HTT
SCHEMBL9221435 0.78 ALDH1A1 (0.56) ALDH1A1CYP3A4MEN1KMT2ACYP1A2
SCHEMBL3183891 0.77 CA12 (0.51) ALDH1A1CYP3A4MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed