SCHEMBL29133435

SCHEMBL29133435

BrCCCCOc1ccc2cccnc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.58
CYP3A4 P08684 1/20 0.57
DRD3 P35462 1/20 0.49
HTT P42858 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C19 P33261 1/20 0.49
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TDP1 Q9NUW8 2/20 0.46
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
KMT2A Q03164 1/20 0.45
NR4A2 P43354 1/20 0.45
GPBAR1 Q8TDU6 1/20 0.44
CYSLTR2 Q9NS75 1/20 0.44
CYSLTR1 Q9Y271 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7068337 0.95 CYP3A4 (0.59) PDE10ACYP3A4DRD3HTTCYP1A2
SCHEMBL14464160 0.90 CYP3A4 (0.60) PDE10ACYP3A4DRD3HTTCYP1A2
SCHEMBL23412137 0.87 CYP3A4 (0.68) PDE10ACYP3A4DRD3HTTCYP1A2
SCHEMBL32667931 0.86 PDE10A (0.60) PDE10ACYP3A4DRD3HTTCYP1A2
SCHEMBL23412263 0.85 NPC1 (0.68) PDE10ACYP3A4DRD3HTTCYP1A2
SCHEMBL30524215 0.85 NPC1 (0.44) PDE10ACYP3A4DRD3HTTNPC1
SCHEMBL28900537 0.84 PDE10A (0.58) PDE10ACYP3A4DRD3HTTCYP1A2
SCHEMBL31238784 0.84 PDE10A (0.58) PDE10ACYP3A4DRD3HTTCYP1A2
SCHEMBL12957491 0.84 CYP3A4 (0.60) PDE10ACYP3A4DRD3HTTCYP1A2
SCHEMBL27976043 0.83 CYP3A4 (0.64) PDE10ACYP3A4DRD3HTTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117327065-A Carbazole derivatives as dopamine D2/3 receptor modulators 北京大学 2024-01-02 CN disclosed
WO-2023143393-A1 TRICYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海科技大学 2023-08-03 WO disclosed
CN-110776459-B Cholinesterase inhibitors of 7-hydroxy-2-quinolone-dithiocarbamates 江苏知原药业股份有限公司 2023-01-24 CN disclosed