SCHEMBL29133722

SCHEMBL29133722

N#Cc1cnc2ccc(-c3cc(Cl)c(O)c(Cl)c3)cc2c1NCCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MELK Q14680 10/20 0.54
MAP3K8 P41279 1/20 0.47
EGFR P00533 4/20 0.44
ABL1 P00519 1/20 0.44
SRC P12931 1/20 0.44
FLT1 P17948 1/20 0.44
KDR P35968 1/20 0.44
SYK P43405 1/20 0.44
PRKDC P78527 2/20 0.43
TNF P01375 1/20 0.43
PIK3CA P42336 1/20 0.43
CCNC P24863 2/20 0.42
CDK8 P49336 2/20 0.42
PDPK1 O15530 1/20 0.42
CDKN1A P38936 1/20 0.42
CDK19 Q9BWU1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133698 0.88 MELK (0.54) MELKMAP3K8EGFRABL1SRC
SCHEMBL29133767 0.84 EGFR (0.44) MELKMAP3K8EGFRABL1SRC
SCHEMBL29133731 0.83 EGFR (0.63) MAP3K8EGFRABL1SRCFLT1
SCHEMBL29133710 0.82 CYP1A2 (0.52) EGFRABL1SRCFLT1KDR
SCHEMBL29133717 0.82 EGFR (0.50) MAP3K8EGFRABL1SRCFLT1
SCHEMBL29133738 0.81 CCNC (0.47) MAP3K8EGFRABL1SRCFLT1
SCHEMBL29133761 0.81 EGFR (0.51) MAP3K8EGFRABL1SRCFLT1
SCHEMBL29133766 0.79 CCNC (0.57) MAP3K8EGFRABL1SRCFLT1
SCHEMBL29133741 0.79 EGFR (0.66) MAP3K8EGFRABL1SRCFLT1
SCHEMBL29133770 0.79 PIK3CA (0.54) EGFRABL1SRCFLT1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117295716-A Substituted aminobenzyl heteroaryl compounds as EGFR and/or PI3K inhibitors 麦克尼斯迪克治疗有限公司 2023-12-26 CN disclosed