SCHEMBL29133741

SCHEMBL29133741

N#Cc1cnc2ccc(-c3cnc4[nH]ncc4c3)cc2c1NCCc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.66
PRKDC P78527 4/20 0.66
SRC P12931 3/20 0.43
ABL1 P00519 1/20 0.43
FLT1 P17948 1/20 0.43
KDR P35968 1/20 0.43
SYK P43405 1/20 0.43
PIK3CA P42336 4/20 0.43
AKT1 P31749 1/20 0.43
CCNC P24863 2/20 0.41
CDK8 P49336 2/20 0.41
CDKN1A P38936 1/20 0.41
CDK19 Q9BWU1 1/20 0.41
MAP3K8 P41279 1/20 0.40
ROCK2 O75116 1/20 0.40
AURKB Q96GD4 1/20 0.40
PDPK1 O15530 1/20 0.40
SLC29A1 Q99808 1/20 0.40
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133717 0.88 EGFR (0.50) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133780 0.88 PIK3CA (0.51) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133709 0.87 EGFR (0.49) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133702 0.84 EGFR (0.49) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133761 0.83 EGFR (0.51) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133731 0.83 EGFR (0.63) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133738 0.82 CCNC (0.47) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133770 0.81 PIK3CA (0.54) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133767 0.81 EGFR (0.44) EGFRPRKDCSRCABL1FLT1
SCHEMBL29133710 0.81 CYP1A2 (0.52) EGFRPRKDCSRCABL1FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117295716-A Substituted aminobenzyl heteroaryl compounds as EGFR and/or PI3K inhibitors 麦克尼斯迪克治疗有限公司 2023-12-26 CN disclosed