SCHEMBL29133780

SCHEMBL29133780

N#Cc1cnc2ccc(-c3cnc4[nH]ccc4c3)cc2c1NCCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.51
MTOR P42345 7/20 0.51
PIK3CD O00329 7/20 0.51
EGFR P00533 4/20 0.51
PRKDC P78527 3/20 0.51
RIPK1 Q13546 1/20 0.46
CDK8 P49336 5/20 0.45
AXL P30530 1/20 0.45
PRKCQ Q04759 1/20 0.44
ABL1 P00519 1/20 0.43
SRC P12931 1/20 0.43
FLT1 P17948 1/20 0.43
KDR P35968 1/20 0.43
SYK P43405 1/20 0.43
TNIK Q9UKE5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133741 0.88 EGFR (0.66) PIK3CAMTORPIK3CDEGFRPRKDC
SCHEMBL29133717 0.88 EGFR (0.50) PIK3CAMTORPIK3CDEGFRPRKDC
SCHEMBL29133709 0.84 EGFR (0.49) PIK3CAEGFRPRKDCCDK8ABL1
SCHEMBL29133702 0.84 EGFR (0.49) PIK3CAMTORPIK3CDEGFRPRKDC
SCHEMBL29133761 0.83 EGFR (0.51) PIK3CAEGFRPRKDCCDK8ABL1
SCHEMBL29133731 0.82 EGFR (0.63) PIK3CAEGFRPRKDCCDK8ABL1
SCHEMBL29133738 0.81 CCNC (0.47) PIK3CAEGFRPRKDCCDK8ABL1
SCHEMBL29133770 0.80 PIK3CA (0.54) PIK3CAMTORPIK3CDEGFRPRKDC
SCHEMBL29133767 0.80 EGFR (0.44) PIK3CAEGFRPRKDCCDK8ABL1
SCHEMBL29133710 0.80 CYP1A2 (0.52) EGFRPRKDCCDK8ABL1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117295716-A Substituted aminobenzyl heteroaryl compounds as EGFR and/or PI3K inhibitors 麦克尼斯迪克治疗有限公司 2023-12-26 CN disclosed