SCHEMBL29135069

SCHEMBL29135069

NC(=O)c1ccc(S(=O)(=O)N2CCCc3ccccc32)cc1.O=C(O)c1ccco1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 0.69
MEN1 O00255 7/20 0.69
LMNA P02545 5/20 0.60
ALDH1A1 P00352 2/20 0.60
HTT P42858 2/20 0.60
TSHR P16473 2/20 0.60
NPSR1 Q6W5P4 1/20 0.60
MAPT P10636 4/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
USP2 O75604 1/20 0.57
GAA P10253 1/20 0.57
PKM P14618 1/20 0.57
AKR1C3 P42330 2/20 0.56
MCL1 Q07820 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
KDM4E B2RXH2 1/20 0.54
HPGD P15428 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29134721 0.89 AKR1C3 (0.70) KMT2AMEN1LMNAALDH1A1HTT
SCHEMBL23559189 0.87 KMT2A (0.81) KMT2AMEN1LMNAALDH1A1HTT
SCHEMBL664021 0.82 KMT2A (1.00) KMT2AMEN1LMNATSHRMAPT
SCHEMBL29134739 0.81 KMT2A (0.70) KMT2AMEN1LMNAALDH1A1HTT
Thiophene Carboxylic Acid SCHEMBL29135071 0.80 KMT2A (0.69) KMT2AMEN1LMNAALDH1A1TSHR
SCHEMBL29134725 0.78 KMT2A (0.65) KMT2AMEN1LMNAALDH1A1TSHR
Benzoic Acid SCHEMBL29134718 0.77 AKR1C3 (0.84) KMT2AMEN1LMNAHTTGAA
SCHEMBL665198 0.77 MEN1 (0.87) KMT2AMEN1LMNAALDH1A1HTT
SCHEMBL5829479 0.75 KMT2A (0.78) KMT2AMEN1LMNAALDH1A1HTT
SCHEMBL10187094 0.74 KMT2A (0.70) KMT2AMEN1LMNAALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117298108-A Androgen receptor and glucocorticoid receptor dual-target inhibitor and application thereof 浙江师范大学 2023-12-29 CN disclosed