SCHEMBL29136004

SCHEMBL29136004

CNC(=O)c1cccc(Cn2cc(CCO)c3cc(-c4cn[nH]c4C(F)(F)F)ccc3c2=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.41
GRK2 P25098 1/20 0.38
MAPK1 P28482 1/20 0.38
TNIK Q9UKE5 1/20 0.37
ROCK2 O75116 2/20 0.36
METAP2 P50579 1/20 0.36
ROCK1 Q13464 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BRD4 O60885 3/20 0.35
GPR52 Q9Y2T5 1/20 0.35
MKNK1 Q9BUB5 2/20 0.35
MKNK2 Q9HBH9 2/20 0.35
CECR2 Q9BXF3 1/20 0.35
TAF1 P21675 1/20 0.35
XDH P47989 1/20 0.34
YTHDC1 Q96MU7 1/20 0.34
DHODH Q02127 1/20 0.34
CYP4F2 P78329 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29779026 1.00 TDO2 (0.41) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL29778614 0.92 TDO2 (0.40) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL29135932 0.92 TDO2 (0.40) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL24616971 0.90 GRK2 (0.40) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL29778679 0.90 GRK2 (0.40) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL29135965 0.90 TDO2 (0.40) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL30656540 0.90 TDO2 (0.40) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL29778506 0.88 TDO2 (0.42) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL24616967 0.88 MAPK1 (0.42) TDO2GRK2MAPK1TNIKROCK2
SCHEMBL29778456 0.88 MAPK1 (0.42) TDO2GRK2MAPK1TNIKROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117136186-A Selective inhibitors of ROCK1 and ROCK2 protein kinases and uses thereof 盖诺斯克公司 2023-11-28 CN claimed
CN-117136186-A Selective inhibitors of ROCK1 and ROCK2 protein kinases and uses thereof 盖诺斯克公司 2023-11-28 CN disclosed