SCHEMBL29136642

SCHEMBL29136642

CC(C)(C)OC(=O)NCc1ccc(CNc2c(N)cnc3ccccc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.48
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
NPC1 O15118 1/20 0.46
GAA P10253 1/20 0.46
RAB9A P51151 1/20 0.46
NAMPT P43490 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GRM5 P41594 1/20 0.43
BRD4 O60885 1/20 0.43
AURKA O14965 1/20 0.42
RPS6KB1 P23443 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
BCHE P06276 1/20 0.40
GRM2 Q14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29947676 1.00 HDAC1 (0.48) HDAC1MEN1KMT2ANPC1GAA
SCHEMBL29947681 0.91 AURKA (0.53) HDAC1MEN1KMT2ANPC1GAA
SCHEMBL29136655 0.91 AURKA (0.53) HDAC1MEN1KMT2ANPC1GAA
SCHEMBL12757192 0.88 MEN1 (0.48) HDAC1MEN1KMT2ANPC1GAA
SCHEMBL1232910 0.87 BCHE (0.52) MEN1KMT2ANPC1GAARAB9A
SCHEMBL204017 0.85 MEN1 (0.48) HDAC1MEN1KMT2ANPC1GAA
SCHEMBL29475728 0.85 BRD4 (0.47) MEN1KMT2ANPC1GAARAB9A
SCHEMBL1034070 0.85 BRD4 (0.47) MEN1KMT2ANPC1GAARAB9A
SCHEMBL1232778 0.85 STK17B (0.47) MEN1KMT2ANPC1GAARAB9A
SCHEMBL30503514 0.85 BRD4 (0.47) MEN1KMT2ANPC1GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355341-A TLR7 and TLR8 agonists for the treatment of cancer and/or infectious diseases 纽约州立大学研究基金会 2024-01-05 CN disclosed