SCHEMBL29136646

SCHEMBL29136646

CC(C)(C)OC(=O)Nc1cccc(CNc2c(N)cnc3ccccc23)c1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 6/20 0.56
RPS6KB1 P23443 5/20 0.56
TOP2A P11388 1/20 0.48
TOP2B Q02880 1/20 0.48
TLR7 Q9NYK1 1/20 0.47
MAP4K4 O95819 1/20 0.42
BRD4 O60885 3/20 0.42
AURKB Q96GD4 2/20 0.42
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
HDAC1 Q13547 1/20 0.40
MET P08581 1/20 0.40
SYK P43405 1/20 0.40
GRM5 P41594 1/20 0.40
PDE4B Q07343 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29947712 1.00 AURKA (0.56) AURKARPS6KB1TOP2ATOP2BTLR7
SCHEMBL29947681 0.89 AURKA (0.53) AURKARPS6KB1TOP2ATOP2BMAP4K4
SCHEMBL29136655 0.89 AURKA (0.53) AURKARPS6KB1TOP2ATOP2BMAP4K4
SCHEMBL29947745 0.85 AURKA (0.51) AURKARPS6KB1TOP2ATOP2BTLR7
SCHEMBL29136627 0.85 AURKA (0.51) AURKARPS6KB1TOP2ATOP2BTLR7
SCHEMBL26981109 0.85 AURKA (0.45) AURKARPS6KB1TOP2ATOP2BAURKB
SCHEMBL29136642 0.84 HDAC1 (0.48) AURKARPS6KB1BRD4MEN1NPC1
SCHEMBL29947676 0.84 HDAC1 (0.48) AURKARPS6KB1BRD4MEN1NPC1
SCHEMBL29136626 0.82 AURKA (0.48) AURKARPS6KB1TOP2ATOP2BTLR7
SCHEMBL29947592 0.82 AURKA (0.48) AURKARPS6KB1TOP2ATOP2BTLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355341-A TLR7 and TLR8 agonists for the treatment of cancer and/or infectious diseases 纽约州立大学研究基金会 2024-01-05 CN disclosed