SCHEMBL29136817

SCHEMBL29136817

CNc1cn2cc(C(C)C)ccc2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 8/20 0.38
CSNK1D P48730 1/20 0.36
CSNK1G2 P78368 1/20 0.36
TP53 P04637 2/20 0.34
KDM4E B2RXH2 2/20 0.34
APP P05067 2/20 0.33
ABL1 P00519 1/20 0.33
MCHR1 Q99705 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
MITF O75030 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KDM5A P29375 1/20 0.32
KDM5C P41229 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
PAX8 Q06710 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PIK3CA P42336 1/20 0.32
NFKB1 P19838 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24834491 0.78 NPC1 (0.52) MAP3K5TP53KDM4EAPPMEN1
SCHEMBL12729862 0.77 MCHR1 (0.39) TP53KDM4EAPPMCHR1MEN1
SCHEMBL798511 0.77 MCHR1 (0.45) TP53KDM4EAPPMCHR1MEN1
Hydrochloric Acid SCHEMBL28842904 0.77 NPC1 (0.50) MAP3K5CSNK1DCSNK1G2TP53KDM4E
SCHEMBL14445622 0.75 MAP3K5 (0.47) MAP3K5ABL1MCHR1PIK3CA
SCHEMBL22479121 0.75 NPC1 (0.33) TP53KDM4EAPPMCHR1MEN1
SCHEMBL28842738 0.75 MAP3K5 (0.52) MAP3K5CSNK1DCSNK1G2TP53KDM4E
SCHEMBL28800311 0.75 PIK3CG (0.55) MAP3K5TP53KDM4EAPPMEN1
SCHEMBL24242318 0.75 MAP3K5 (0.36) MAP3K5CSNK1DCSNK1G2TP53KDM4E
SCHEMBL26432426 0.75 KDM4E (0.58) MAP3K5TP53KDM4EAPPABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed