SCHEMBL29137029

SCHEMBL29137029

Nc1cc(Cl)cc(/C=C/C(=O)O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.56
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44
HDAC11 Q96DB2 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44
HDAC5 Q9UQL6 2/20 0.44
HCAR2 Q8TDS4 2/20 0.44
TNKS O95271 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
CYP3A4 P08684 2/20 0.43
ITGB2 P05107 1/20 0.43
ICAM1 P05362 1/20 0.43
ITGAL P20701 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1251510 0.86 HDAC3 (0.52) NPSR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL28774295 0.86 NPSR1 (0.66) NPSR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL1251511 0.86 HDAC3 (0.52) NPSR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL28774292 0.86 NPSR1 (0.66) NPSR1HDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL6818359 0.84 HDAC3 (0.50) NPSR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL29136758 0.80 TTR (0.47) HCAR2CYP3A4TP53KDM4EHSD17B10
SCHEMBL29879341 0.80 TTR (0.47) HCAR2CYP3A4TP53KDM4EHSD17B10
SCHEMBL29136808 0.80 TTR (0.47) HCAR2CYP3A4TP53KDM4EHSD17B10
SCHEMBL4716668 0.78 HDAC3 (0.44) NPSR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL4716666 0.78 HDAC3 (0.44) NPSR1HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed