SCHEMBL29137075

SCHEMBL29137075

COC(=O)C=Cc1cc(Cl)cc(NC(=O)OC(C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
EGFR P00533 1/20 0.40
TTR P02766 1/20 0.40
APP P05067 1/20 0.40
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA9 Q16790 3/20 0.39
CA2 P00918 2/20 0.39
TYR P14679 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
PTPN1 P18031 1/20 0.38
EPHX2 P34913 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
JAK2 O60674 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29302330 1.00 HDAC3 (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL29137052 0.88 HDAC3 (0.44) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL3928304 0.85 BACE1 (0.48) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL3928300 0.85 BACE1 (0.48) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL29953301 0.82 CA12 (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12527219 0.82 CA12 (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL3786493 0.80 L3MBTL1 (0.44) CA12CA1CA9ALDH1A1MAPT
SCHEMBL5879121 0.80 L3MBTL1 (0.47) CA12CA1CA9ALDH1A1MAPT
SCHEMBL5701010 0.80 CA12 (0.55) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL5701011 0.80 CA12 (0.55) HDAC3HDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed