SCHEMBL29137932

SCHEMBL29137932

CC(C)(C)OC(=O)Nc1cc2cc(F)cc(CO)c2cn1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.44
DYRK1A Q13627 1/20 0.44
MAP4K1 Q92918 12/20 0.39
CDK9 P50750 1/20 0.38
SYK P43405 1/20 0.37
MAPK1 P28482 2/20 0.37
GRM2 Q14416 1/20 0.36
MAPKAPK2 P49137 1/20 0.35
TSHR P16473 1/20 0.35
FSHR P23945 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14904853 0.83 GSK3B (0.47) GSK3BDYRK1AMAP4K1CDK9SYK
SCHEMBL20647996 0.82 GSK3B (0.44) GSK3BDYRK1ACDK9SYKMAPK1
SCHEMBL29703975 0.82 GSK3B (0.44) GSK3BDYRK1ACDK9SYKMAPK1
SCHEMBL29137922 0.82 GSK3B (0.41) GSK3BDYRK1AMAP4K1CDK9SYK
SCHEMBL29874548 0.77 GRM2 (0.35) SYKGRM2
SCHEMBL14904903 0.76 GSK3B (0.47) GSK3BDYRK1ACDK9SYKMAPK1
SCHEMBL20520009 0.75 GSK3B (0.47) GSK3BDYRK1AMAP4K1CDK9SYK
SCHEMBL29703935 0.75 SCN9A (0.40) GSK3BDYRK1ACDK9SYKGRM2
SCHEMBL30636312 0.74 GRM2 (0.35) SYKGRM2
SCHEMBL26933292 0.74 GRM2 (0.35) SYKGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117062804-A 1, 3-substituted cyclobutyl derivatives and their use 诺华股份有限公司 2023-11-14 CN disclosed