SCHEMBL29137922

SCHEMBL29137922

CC(C)(C)OC(=O)Nc1cc2cc(F)cc(C(O)CO)c2cn1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
MAPK1 P28482 5/20 0.37
MAP4K1 Q92918 6/20 0.37
CDK9 P50750 1/20 0.36
SYK P43405 1/20 0.35
SCN9A Q15858 1/20 0.35
ABL1 P00519 3/20 0.34
MAPKAPK2 P49137 1/20 0.33
TSHR P16473 1/20 0.33
FSHR P23945 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29137932 0.82 GSK3B (0.44) GSK3BDYRK1AMAPK1MAP4K1CDK9
SCHEMBL29874252 0.79 PDPK1 (0.33) SYK
SCHEMBL30636388 0.77 GRM2 (0.33) SYK
SCHEMBL20520009 0.72 GSK3B (0.47) GSK3BDYRK1AMAPK1MAP4K1CDK9
SCHEMBL20778049 0.71 GSK3B (0.44) GSK3BDYRK1AMAPK1CDK9SYK
SCHEMBL20647996 0.71 GSK3B (0.44) GSK3BDYRK1AMAPK1CDK9SYK
SCHEMBL29703975 0.71 GSK3B (0.44) GSK3BDYRK1AMAPK1CDK9SYK
SCHEMBL14904853 0.70 GSK3B (0.47) GSK3BDYRK1AMAPK1MAP4K1CDK9
SCHEMBL12724232 0.70 CDK9 (0.44) GSK3BDYRK1ACDK9SYKABL1
SCHEMBL29137954 0.70 SCN9A (0.35) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117062804-A 1, 3-substituted cyclobutyl derivatives and their use 诺华股份有限公司 2023-11-14 CN disclosed