SCHEMBL29139939

SCHEMBL29139939

CCCCCCC(CC)c1ccccc1C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 2/20 0.49
PRSS2 P07478 1/20 0.49
PRSS3 P35030 1/20 0.49
ALDH1A1 P00352 4/20 0.45
TSHR P16473 3/20 0.43
LMNA P02545 2/20 0.43
CYP3A4 P08684 2/20 0.42
CA2 P00918 1/20 0.42
CYSLTR2 Q9NS75 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CTSG P08311 1/20 0.39
CTRB1 P17538 1/20 0.39
CMA1 P23946 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30768235 0.91 PRSS1 (0.44) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL28479311 0.86 PRSS1 (0.45) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL29139948 0.85 PRSS1 (0.52) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL28532492 0.85 PRSS1 (0.52) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL6479756 0.84 PRSS1 (0.50) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL29148911 0.84 PRSS1 (0.50) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL671032 0.81 ALDH1A1 (0.55) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL1586807 0.81 PRSS1 (0.53) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL30479012 0.80 CYP3A4 (0.51) PRSS1PRSS2PRSS3ALDH1A1TSHR
SCHEMBL27199692 0.80 CYP3A4 (0.51) PRSS1PRSS2PRSS3ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683029-A Bcl-2 inhibitors 百济神州有限公司 2024-03-12 CN disclosed
CN-117430601-A Bcl-2 inhibitors 百济神州有限公司 2024-01-23 CN disclosed
CN-112437772-B Bcl-2 inhibitors 百济神州有限公司 2023-11-21 CN disclosed