SCHEMBL29142175

SCHEMBL29142175

COc1ccc(CNc2ncccc2C2(NC(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
KLKB1 P03952 4/20 0.42
F2 P00734 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ASPH Q12797 1/20 0.41
KDM8 Q8N371 1/20 0.41
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CDK5 Q00535 3/20 0.39
CDK5R1 Q15078 3/20 0.39
AURKA O14965 1/20 0.39
RPS6KB1 P23443 1/20 0.39
KLK1 P06870 1/20 0.39
ALDH1A1 P00352 3/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27088549 0.79 NPC1 (0.49) NPC1KDM4EASPHKDM8MEN1
SCHEMBL29142207 0.78 NPC1 (0.51) NPC1KLKB1F2KDM4EASPH
SCHEMBL27478229 0.75 AKT1 (0.46) RAB9APOLB
SCHEMBL29999288 0.75 NPC1 (0.40) NPC1KLKB1F2KDM4EASPH
SCHEMBL27088912 0.74 POLB (0.44) KDM4ELMNASMN1; SMN2RAB9APOLB
SCHEMBL30518086 0.74 FFAR1 (0.41) NPC1KDM4EASPHKDM8MEN1
SCHEMBL25155751 0.73 AKT1 (0.42) NPC1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL31360275 0.73 AKT1 (0.42) NPC1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL30344108 0.73 AKT1 (0.42) NPC1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL1715769 0.73 NPC1 (0.66) NPC1KLKB1KDM4EASPHKDM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117083279-A Oxazepine compounds and their use in the treatment of cancer 基因泰克公司 2023-11-17 CN disclosed