SCHEMBL2914800

SCHEMBL2914800

CN(C(=O)O)[C@@H]1CCCC(c2c[nH]c3ccc(NC(=N)c4cccs4)cc23)C1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.47
NOS3 P29474 11/20 0.47
NOS1 P29475 11/20 0.47
NOS2 P35228 9/20 0.47
KCNH2 Q12809 6/20 0.47
CYP3A4 P08684 5/20 0.47
CYP2D6 P10635 5/20 0.47
HTR1B P28222 5/20 0.42
HTR1D P28221 4/20 0.42
HTR1A P08908 2/20 0.42
HTR1F P30939 1/20 0.42
CYP2C19 P33261 4/20 0.41
CYP2C9 P11712 2/20 0.41
SLC6A4 P31645 5/20 0.41
DRD1 P21728 1/20 0.41
HTR2A P28223 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2908452 1.00 SLC6A2 (0.47) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL1122007 0.91 NOS3 (0.52) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL2911117 0.89 NOS3 (0.47) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL13776968 0.89 SLC6A2 (0.43) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL2919909 0.85 SLC6A2 (0.45) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL2263052 0.83 NOS3 (0.46) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL2931173 0.83 NOS3 (0.66) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL4143576 0.83 NOS3 (0.66) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL13846453 0.83 NOS3 (0.51) SLC6A2NOS3NOS1NOS2KCNH2
SCHEMBL13846432 0.82 NOS3 (0.49) SLC6A2NOS3NOS1NOS2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220074-A1 3,5-SUBSTITUTED INDOLE COMPOUNDS HAVING NOS AND NOREPINEPHRINE REUPTAKE INHIBITORY ACTIVITY Neuraxon, INC. (CA) 2010-08-25 EP disclosed
WO-2009062318-A1 3,5-SUBSTITUTED INDOLE COMPOUNDS HAVING NOS AND NOREPINEPHRINE REUPTAKE INHIBITORY ACTIVITY NEURAXON, INC. (CA) 2009-05-22 WO disclosed