SCHEMBL29149059

SCHEMBL29149059

COc1cc2cccc(C)c2n1C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 15/20 0.41
NR1H3 Q13133 3/20 0.37
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
GPR119 Q8TDV5 1/20 0.34
BCHE P06276 1/20 0.34
BACE1 P56817 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31462830 0.82 NR1H2 (0.43) NR1H2NR1H3
SCHEMBL19013553 0.82 NR1H2 (0.40) NR1H2NR1H3CA12CA9
SCHEMBL29631893 0.82 NR1H2 (0.40) NR1H2NR1H3CA12CA9
SCHEMBL15528336 0.81 PLA2G10 (0.36) CA12CA9
SCHEMBL30933380 0.81 PLA2G10 (0.36) CA12CA9
SCHEMBL13515301 0.80 NR1H2 (0.40) NR1H2NR1H3CA12CA9GPR119
SCHEMBL19013505 0.80 NR1H2 (0.43) NR1H2NR1H3CA12CA9GPR119
SCHEMBL28370896 0.79 NR1H2 (0.55) NR1H2NR1H3CA12CA9
SCHEMBL15431762 0.76 BACE1 (0.43) NR1H2NR1H3CA12CA9BACE1
SCHEMBL30721531 0.73 NQO2 (0.48) NR1H2NR1H3BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118043314-A Benzazepine heteroaromatic ring derivative and application thereof in medicine 西藏海思科制药有限公司 2024-05-14 CN disclosed
CN-117500499-A Substituted indole compounds and methods of use thereof 奇努克治疗公司 2024-02-02 CN disclosed
WO-2023246677-A1 INDOLE-PHENYLPIPERIDINE COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF 深圳信立泰药业股份有限公司 2023-12-28 WO disclosed