SCHEMBL29149554

SCHEMBL29149554

O=C1CCC(C(=O)Nc2cc(OC3CCC(F)(F)CC3)cc3c2OCC3)CN1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
SLC5A1 P13866 11/20 0.36
RXFP1 Q9HBX9 1/20 0.35
IP6K1 Q92551 1/20 0.35
IP6K3 Q96PC2 1/20 0.35
IP6K2 Q9UHH9 1/20 0.35
CDK9 P50750 1/20 0.34
RORC P51449 1/20 0.33
KDM1A O60341 1/20 0.33
ACACB O00763 1/20 0.33
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29938542 1.00 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DSLC5A1
SCHEMBL24750189 0.89 SLC5A1 (0.36) PDE4APDE4BPDE4CPDE4DSLC5A1
SCHEMBL24749754 0.77 RXFP1 (0.37) PDE4APDE4BPDE4CPDE4DRXFP1
SCHEMBL29149358 0.73 SCN9A (0.49) SLC5A1
SCHEMBL24749710 0.71 RXFP1 (0.34) PDE4APDE4BPDE4CPDE4DRXFP1
SCHEMBL31009381 0.71 RXFP1 (0.34) PDE4APDE4BPDE4CPDE4DRXFP1
SCHEMBL24749658 0.71 RXFP1 (0.34) PDE4APDE4BPDE4CPDE4DRXFP1
Hydrochloric Acid SCHEMBL31694844 0.70 RXFP1 (0.33) PDE4APDE4BPDE4CPDE4DRXFP1
SCHEMBL24749996 0.66 P2RX7 (0.33) KDM1A
SCHEMBL29938408 0.66 P2RX7 (0.33) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117500786-A TEAD inhibitors 奥赖恩公司 2024-02-02 CN disclosed