Thiophene Carboxylic Acid

Thiophene Carboxylic Acid

SCHEMBL2915010

NC(=O)O.O=C(O)c1cccs1

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.86
CES2 O00748 1/20 0.60
CES1 P23141 1/20 0.60
HPGDS O60760 1/20 0.55
LMNA P02545 3/20 0.55
ALOX15 P16050 1/20 0.55
KMT2A Q03164 6/20 0.54
MEN1 O00255 5/20 0.54
RAB9A P51151 4/20 0.54
NPC1 O15118 3/20 0.54
ALDH1A1 P00352 1/20 0.54
POLB P06746 1/20 0.54
HDAC1 Q13547 1/20 0.54
HPGD P15428 3/20 0.50
GSK3B P49841 1/20 0.50
NOS1 P29475 1/20 0.50
PKM P14618 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HTT P42858 1/20 0.50
ERCC5 P28715 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiophene Carboxylic Acid SCHEMBL9134447 0.93 DAO (0.91) DAOCES2CES1HPGDSLMNA
Thiophene Carboxylic Acid SCHEMBL7062244 0.93 DAO (1.00) DAOCES2CES1HPGDSLMNA
Thiophene Carboxylic Acid SCHEMBL83000 0.93
Thiophene Carboxylic Acid SCHEMBL27774764 0.93 DAO (1.00) DAOCES2CES1HPGDSLMNA
Thiophene Carboxylic Acid SCHEMBL7263058 0.91 DAO (0.86) DAOCES2CES1HPGDSLMNA
Thiophene Carboxylic Acid SCHEMBL5287669 0.91 DAO (0.95) DAOCES2CES1HPGDSLMNA
Thiophene Carboxylic Acid SCHEMBL1814 0.91
Thiophene Carboxylic Acid SCHEMBL20895852 0.91
Thiophene Carboxylic Acid SCHEMBL4331473 0.91
Thiophene Carboxylic Acid SCHEMBL10898170 0.91

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1438073-B1 POLYOXYALKYLENE CONJUGATES AS ENZYME INHIBITORS PROCTER & GAMBLE (US) 2010-08-11 EP disclosed
EP-1438073-A2 POLYOXYALKYLENES CONJUGATES AS ENZYME INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2004-07-21 EP disclosed
US-6723788-B1 Enzyme inhibitors THE PROCTER & GAMBLE COMPANY 2004-04-20 US disclosed
US-6541629-B1 An enzyme inhibitor containing benzoxazine ring attached with 1-16 ethoxy groups used for treating diaper rash THE PROCTER & GAMBLE COMPANY 2003-04-01 US disclosed
EP-1212097-A2 ENZYME INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2002-06-12 EP disclosed
EP-1212098-A2 ENZYME INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2002-06-12 EP disclosed
WO-2001017564-A2 ENZYME INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2001-03-15 WO disclosed
WO-2001017565-A2 POLYOXYALKYLENES CONJUGATES AS ENZYME INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2001-03-15 WO disclosed
WO-2001018181-A2 ENZYME INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2001-03-15 WO disclosed