SCHEMBL29164181

SCHEMBL29164181

COc1ccc(Cl)c(Cl)c1[C@@H]1CCC(CO)N1C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.44
HTR2C P28335 6/20 0.44
HTR2B P41595 6/20 0.44
PDE4B Q07343 7/20 0.38
DRD2 P14416 1/20 0.37
PDE4A P27815 3/20 0.36
PDE4C Q08493 3/20 0.36
PDE4D Q08499 3/20 0.36
STS P08842 1/20 0.35
OPRK1 P41145 1/20 0.34
SUV39H2 Q9H5I1 1/20 0.34
FFAR2 O15552 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29164179 1.00 HTR2A (0.44) HTR2AHTR2CHTR2BPDE4BDRD2
SCHEMBL30721093 1.00 HTR2A (0.44) HTR2AHTR2CHTR2BPDE4BDRD2
SCHEMBL29164180 0.89 HTR2A (0.45) HTR2AHTR2CHTR2BPDE4BDRD2
SCHEMBL30721087 0.89 HTR2A (0.45) HTR2AHTR2CHTR2BPDE4BDRD2
SCHEMBL29164183 0.89 HTR2A (0.45) HTR2AHTR2CHTR2BPDE4BDRD2
SCHEMBL30721060 0.88 HTR2A (0.41) HTR2AHTR2CHTR2BPDE4BDRD2
SCHEMBL29164185 0.88 HTR2A (0.41) HTR2AHTR2CHTR2BPDE4BDRD2
SCHEMBL29164189 0.88 HTR2A (0.41) HTR2AHTR2CHTR2BPDE4BDRD2
SCHEMBL30120779 0.86 HTR2A (0.45) HTR2AHTR2CHTR2BDRD2FFAR2
SCHEMBL30721081 0.83 ALDH1A1 (0.43) HTR2AHTR2CHTR2BPDE4BPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117337280-A Aryl heterocyclic compounds as Kv1.3 potassium SHAKER channel blockers D·E·萧尔研究有限责任公司 2024-01-02 CN disclosed