Oxirane

Oxirane

SCHEMBL29170802

C1CO1.Cc1ccncc1Br

nearest known ligand 0.37

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT3 Q9NTG7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
OPRL1 P41146 2/20 0.35
ALDH1A1 P00352 3/20 0.34
PIK3C3 Q8NEB9 1/20 0.34
CYP1A2 P05177 4/20 0.33
CYP2E1 P05181 3/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2C8 P10632 3/20 0.33
CYP2D6 P10635 3/20 0.33
CYP2A6 P11509 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP2B6 P20813 3/20 0.33
CYP2C19 P33261 3/20 0.33
AXL P30530 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
CYP17A1 P05093 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29720188 0.89
SCHEMBL314379 0.89
Hydrochloric Acid SCHEMBL27912104 0.87
Cyanide SCHEMBL27862175 0.83 SIRT3 (0.39) SIRT3TDP1IDO1TDO2ALDH1A1
Formaldehyde SCHEMBL29175656 0.83 SIRT3 (0.44) SIRT3TDP1IDO1TDO2ALDH1A1
SCHEMBL793800 0.74
SCHEMBL29741232 0.70
SCHEMBL550773 0.70
Ethoxycarbonyl Group SCHEMBL27884564 0.70 CA12 (0.36) SIRT3TDP1CYP1A2CYP2E1CYP3A4
Hydrochloric Acid SCHEMBL25411609 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117447475-A Pyrazolo [4,3-b ] pyridines and imidazo [1,5-a ] pyrimidines as PDE1 inhibitors H.隆德贝克有限公司 2024-01-26 CN disclosed