SCHEMBL29176282

SCHEMBL29176282

COc1ccc(-c2cc3c(cn2)n(CC(N)=O)c(=O)n3-c2cc(OC)c(OC)c(OC)c2)cc1OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.49
ABCB1 P08183 3/20 0.46
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 3/20 0.44
KATNA1 O75449 1/20 0.40
MAPT P10636 1/20 0.40
PDE4A P27815 4/20 0.40
PDE4B Q07343 4/20 0.40
PDE4C Q08493 4/20 0.40
PDE4D Q08499 4/20 0.40
PDE5A O76074 2/20 0.39
MAPK1 P28482 1/20 0.39
SMPD1 P17405 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30800025 1.00 SMN1; SMN2 (0.49) SMN1; SMN2ABCB1KMT2AMEN1ALDH1A1
SCHEMBL30800052 0.87 TSHR (0.45) SMN1; SMN2ABCB1KMT2AMEN1ALDH1A1
SCHEMBL29176270 0.87 TSHR (0.45) SMN1; SMN2ABCB1KMT2AMEN1ALDH1A1
SCHEMBL30799997 0.86 KATNA1 (0.54) SMN1; SMN2KMT2AMEN1ALDH1A1LMNA
SCHEMBL29176273 0.86 KATNA1 (0.54) SMN1; SMN2KMT2AMEN1ALDH1A1LMNA
SCHEMBL30799993 0.84 ABCB1 (0.43) SMN1; SMN2ABCB1KMT2AKATNA1PDE4A
SCHEMBL29176310 0.84 ABCB1 (0.43) SMN1; SMN2ABCB1KMT2AKATNA1PDE4A
SCHEMBL29176300 0.79 KATNA1 (0.47) SMN1; SMN2ABCB1KMT2AKATNA1PDE4A
SCHEMBL30799992 0.79 KATNA1 (0.47) SMN1; SMN2ABCB1KMT2AKATNA1PDE4A
SCHEMBL29176287 0.75 KATNA1 (0.50) SMN1; SMN2KMT2AMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111732584-B Diaryl substituted fused heterocycle compound and preparation method and application thereof in pharmacy 复旦大学 2024-02-27 CN disclosed