SCHEMBL30799993

SCHEMBL30799993

COc1ccc(-c2cc3c(cn2)n(C(=O)C2CC2)c(=O)n3-c2cc(OC)c(OC)c(OC)c2)cc1OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PKM P14618 1/20 0.40
PDCD1 Q15116 2/20 0.39
CD274 Q9NZQ7 2/20 0.39
KMT2A Q03164 1/20 0.38
KATNA1 O75449 1/20 0.38
SMPD1 P17405 2/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
APP P05067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29176310 1.00 ABCB1 (0.43) ABCB1SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL29176282 0.84 SMN1; SMN2 (0.49) ABCB1SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL30800025 0.84 SMN1; SMN2 (0.49) ABCB1SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL30800052 0.82 TSHR (0.45) ABCB1SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL29176270 0.82 TSHR (0.45) ABCB1SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL30799992 0.77 KATNA1 (0.47) ABCB1SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL29176300 0.77 KATNA1 (0.47) ABCB1SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL29176291 0.72 MAP3K11 (0.48) ABCB1PDE4APDE4BPDE4CPDE4D
SCHEMBL30800080 0.72 MAP3K11 (0.48) ABCB1PDE4APDE4BPDE4CPDE4D
SCHEMBL28474690 0.71 KATNA1 (0.49) PDE4APDE4BPDE4CPDE4DKATNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111732584-B Diaryl substituted fused heterocycle compound and preparation method and application thereof in pharmacy 复旦大学 2024-02-27 CN disclosed